當(dāng)前位置：珀金埃爾默醫(yī)學(xué)診斷產(chǎn)品（上海）有限公司>>>>Diltiazem, cis-(+)-[N-Methyl-3H]-, 250µCi (9.25MBq)

Diltiazem, cis-(+)-[N-Methyl-3H]-, 250µCi (9.25MBq)

返回列表頁

參考價

面議

具體成交價以合同協(xié)議為準(zhǔn)

產(chǎn)品型號

品牌

廠商性質(zhì)其他

所在地

在線詢價收藏產(chǎn)品查看聯(lián)系電話

聯(lián)系方式：查看聯(lián)系方式

更新時間：2022-10-12 13:05:25瀏覽次數(shù)：97次

聯(lián)系我時，請告知來自環(huán)保在線

產(chǎn)品分類 品牌分類

暫無信息

珀金埃爾默醫(yī)學(xué)診斷產(chǎn)品（上海）有限公司

經(jīng)營模式：其他

商鋪產(chǎn)品：677條

所在地區(qū)：

詢價 給他留言

產(chǎn)品簡介

cis-(+)-Diltiazem, tritiated at the N-methyl position. Diltiazem is a non-DHP calcium channel blocker.

詳細(xì)介紹

Diltiazem is a nondihydropyridine (non-DHP) calcium channel blocker used to treat hypertension and arrythmia.

We offer both agonist and antagonist radioligands for autoradiographic visualization or performing saturation and competition assays to determine receptor expression levels (B_max), dissociation constants (K_d), association and dissociation rates (k_on and k_off), and inhibitor constants (K_i) for a variety of receptors. We develop our radioligands to the highest specific activity possible and provide high purity resulting in low non-specific binding products. Each of our ultra-pure radioligands is fully characterized for pharmacological action and validated in receptor binding assays.

Radiolabeled ligands remain the most sensitive method for probing receptor binding biology; yielding unprecedented sensitivity gives results that technicians and scientists can trust. For over 50 years, PerkinElmer has been a leading supplier of New Englａnd Nuclear (NEN) radiochemicals, liquid scintillation cocktails, vials and nuclear counting detection instruments.

References for NET847:

Rupniak, N.M.J., Boyce, S., Williams, A.R., Cook, G., Longmore, J., Seabrook, G.R., Caeser, M., Iversen, S.D. and Hill, R.G. (1993), Antinociceptive activity of NK1 receptor antagonists: non-specific effects of racemic RP67580. British Journal of Pharmacology, 110: 1607–1613.
Hans Schoemaker, Polyamines allosterically modulate [3H]nitrendipine binding to the voltage-sensitive calcium channel in rat brain, In European Journal of Pharmacology: Molecular Pharmacology, Volume 225, Issue 2, 1992, Pages 167-169.

規(guī)格

濃度	1.0 - 10 mCi/mL
檢測方法	Radiometric
標(biāo)簽位置	Specifically Labeled
分子量	414.5
產(chǎn)品品牌名稱	NEN Radiochemicals
放射性同位素	H-3
放射性核素	³H
受體類型	Calcium
運(yùn)輸條件	干冰
特殊訂購信息	This is a radioactive product - shipping address must have a license to receive radioactive materials.
治療領(lǐng)域	CNS & Neurologic, Pain
產(chǎn)品尺寸	250 µCi